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IL-23R

요약

Name:Interleukin 23 Receptor
Target Synonym:IL-23 receptor,IL23R,Interleukin 23 Receptor,Interleukin-23 Receptor,IL-23R
Number of Launched Drugs:1
Number of Drugs in Clinical Trials:3
Lastest Research Phase:Approved

제품 리스트 구매

일부의 생물활성 데이터

ILR-H5254-SPR
 IL-23R SPR

Captured Human IL-23 R, Fc Tag (Cat. No. ILR-H5254) on CM5 chip via anti-human IgG Fc antibodies surface can bind Human IL23A & IL12B, His Tag (Cat. No. ILB-H52W5)with an affinity constant of 5.36 nM as determined in a SPR assay (Biacore T200) (Routinely tested).

ILR-H52H4-SPR
 IL-23R SPR

Biotinylated Human IL-23A&IL-12B Heterodimer Protein, His,Avitag&Tag Free (Cat. No. ILB-H82W6) captured on Biotin CAP - Series S sensor Chip can bind Human IL-23 R, His Tag (SPR verified) (Cat. No. ILR-H52H4) with an affinity constant of 3.39 nM as determined in a SPR assay (Biacore 8K) (QC tested).

Synonym Name

IL-23 R,IL-23 Receptor

Background

Interleukin 23 receptor (IL-23R) is a type I cytokine receptor, and IL-23R pairs with the receptor molecule IL12RB1/IL12Rbeta1, and both are required for IL23A signaling. Also, IL-23R associates constitutively with Janus kinase 2 (JAK2), and binds to transcription activator STAT3 in a ligand-dependent manner. Furthermore, IL-23R mediates T-cells, NK cells and possibly certain macrophage/myeloid cells stimulation probably through activation of the Jak-Stat signaling cascade. As for IL-23, it may be responsible for autoimmune inflammatory diseases and be important for tumorigenesis.

Clinical and Translational Updates

공개 약품 정보

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Ustekinumab biosimilar (Samsung Bioepis) SB-17; SB17 Approved Samsung Bioepis Co Ltd Pyzchiva EU Crohn Disease; Colitis, Ulcerative Samsung Bioepis Nl Bv 2024-04-19 Gastrointestinal Diseases; Skin Diseases; Psoriasis; Colitis, Ulcerative; Arthritis, Psoriatic; Rheumatic Diseases; Inflammation; Crohn Disease; Plaque psoriasis Details

임상 약품 정보

Name Research Code Research Phase Company Indications Clinical Trials
Bezisterim HE-3286; NE-3107 Phase 3 Clinical Harbor Therapeutics, Biovie Inc Diabetes Mellitus, Type 2; Brain Injuries, Traumatic; Insulin Resistance; Arthritis, Rheumatoid; Post-Acute COVID-19 Syndrome; Alzheimer Disease; Parkinson Disease; Colitis, Ulcerative Details
Icotrokinra PN-235; JNJ-2113; PN-21235; JNJ-77242113-AAC; JNJ-77242113 Phase 3 Clinical Protagonist Therapeutics Inc Psoriasis; Arthritis, Psoriatic; Colitis, Ulcerative; Plaque psoriasis Details
PN-232 PN-232; JNJ75105186 Phase 1 Clinical Protagonist Therapeutics Inc Details

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