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Your Position: > Integrin alpha V beta 3

Integrin alpha V beta 3

요약

Name:Integrin alpha-V/beta-3
Target Synonym:Integrin alphaVbeta3
Number of Launched Drugs:0
Number of Drugs in Clinical Trials:25
Lastest Research Phase:NDA/BLA

제품 리스트 구매

일부의 생물활성 데이터

IT3-H52E3-SPR
 Integrin alpha V beta 3 SPR

Human EDIL3, Fc Tag (Cat. No. ED3-H5259) immobilized on CM5 Chip can bind Human ITGAV&ITGB3 Heterodimer Protein, His Tag&Tag Free (Cat. No. IT3-H52E3) with an affinity constant of 38.9 nM as determined in a SPR assay (Biacore 8K) (Routinely tested).

IT3-R52E2-ELISA
 Integrin alpha V beta 3 ELISA

Immobilized Human Vitronectin at 5 μg/mL (100 μL/well) can bind Rat ITGAV&ITGB3 Heterodimer, His Tag&Tag Free (Cat. No. IT3-R52E2) with a linear range of 0.039-1.25 μg/mL (QC tested).

Synonym Name

Integrin alpha V beta 3,ITGAV&ITGB3

Background

Integrin alpha-V/beta-3 (ITGAV:ITGB3) is a receptor for cytotactin, fibronectin, laminin, matrix metalloproteinase-2, osteopontin, osteomodulin, prothrombin, thrombospondin, vitronectin and von Willebrand factor. Integrins alpha-IIb/beta-3 and alpha-V/beta-3 recognize the sequence R-G-D in a wide array of ligands. Also, Integrin alpha-V/beta-3 acts as a receptor for herpes virus 8/HHV-8, coxsackievirus A9, Hantaan virus, cytomegalovirus/HHV-5, human metapneumovirus, human parechovirus 1 and west nile virus. Furthermore, in case of HIV-1 infection, the interaction with extracellular viral Tat protein seems to enhance angiogenesis in Kaposi's sarcoma lesions.

Clinical and Translational Updates

임상 약품 정보

Name Research Code Research Phase Company Indications Clinical Trials
Alfatide[18F] 18F-AlF-NOTA-PRGD2; 18F-alfatide; alfatide II; AlF-NOTA-PRGD2-[18F] Phase 3 Clinical Jiangsu Smk Pharmaceutical Co Ltd, Taizhou Kairui Pharmaceutical Technology Co Ltd Head and Neck Neoplasms; Carcinoma, Bronchogenic; Neoplasms; Soft Tissue Neoplasms; Breast Neoplasms; Contrast agents; Lymphoma; Lung Neoplasms; Carcinoma, Non-Small-Cell Lung Details
18F-LNC1016 18F-LNC1016; 18F-LNC-1016 Phase 3 Clinical Shanghai Lannacheng Biotechnology Co Ltd Lung Neoplasms Details
IDL-2965 IDL-2965 Phase 2 Clinical Indalo Therapeutics Inc Metabolic Dysfunction-Associated Steatotic Liver Disease; Idiopathic Pulmonary Fibrosis Details
AS-101 PRX-0001/AS101; WAX-120337; IVAX-Q-101; IVX-Q-101; CB-06-02; AS-101; PRX-001; PRX-0002/AS101 Phase 2 Clinical Biomas Ltd HIV Infections; Alopecia; Warts; Myelodysplastic Syndromes; Psoriasis; Leukemia, Myeloid, Acute; Thrombocytopenia; Condylomata Acuminata; Dermatitis, Atopic; Macular Degeneration Details
Nesvategrast OTT-166(OcuTerra Therapeutics); SF-0166 Phase 2 Clinical Scifluor Life Sciences Inc, OcuTerra Therapeutics Inc Diabetic macular oedema; Diabetic Retinopathy; Macular Degeneration Details
ProAgio Phase 2 Clinical National Cancer Institute Solid tumours; Pancreatic Neoplasms; Triple Negative Breast Neoplasms Details
Ga-68 NODAGA-RGD [68Ga]Theranost; Theranost 68Ga-RGD Phase 1 Clinical Advanced Imaging Projects, Zentralklinik Bad Berka, National Cancer Institute Neovascularization, Pathologic; Lung Neoplasms Details
Risuteganib ALG-1001; AM011; AM-011(Allegro Ophthalmics) Phase 1 Clinical Allegro Ophthalmics Llc Diabetic macular oedema; Geographic Atrophy; Diabetic Retinopathy; Macular Degeneration Details
68Ga-NOTA-BBN-RGD 68Ga-NOTA-BBN-RGD Phase 1 Clinical Peking Union Medical College Hospital Breast Neoplasms; Prostatic Neoplasms Details
BGC-0222 BGC0222; BGC-0222 Phase 1 Clinical Gaorui Yaoye (Beijing) Technologies Co Ltd, Brightgene Bio-Medical Technology Co Ltd Solid tumours Details
Antiangiotide HM-3; IIM-3 Phase 1 Clinical Inner Mongolia Tianqi Pharmaceutical Group Co Ltd, China Pharmaceutical University Liver Neoplasms; Solid tumours; Stomach Neoplasms; Carcinoma, Non-Small-Cell Lung Details
68Ga-NOTA-3PTATE-RGD 68Ga-NOTA-3PTATE-RGD; 68Ga-NOTA-3P-TATE-RGD Phase 1 Clinical Peking Union Medical College Hospital Neuroendocrine Tumors; Lung Neoplasms; Meningioma Details
FF-10158 FF-10158 Phase 1 Clinical Fujifilm Holdings Corp Glioblastoma Details
Transferrin OCU-200 Phase 1 Clinical Ocugen Inc Wet Macular Degeneration; Diabetic macular oedema; Diabetic Retinopathy Details
VIP-236 VIP-236 Phase 1 Clinical Bayer AG Solid tumours; Neoplasms Details
177Lu-FAPI-RGD 177Lu-FAPI-RGD Phase 1 Clinical Peking Union Medical College Hospital Neoplasms Details
177Lu-LNC1008 177Lu-LNC1008 Phase 1 Clinical Shanghai Lannacheng Biotechnology Co Ltd Solid tumours Details
68Ga-FAPI-RGD 68Ga-FAPI-RGD; 68Ga-LNC-1007 Phase 1 Clinical Peking Union Medical College Hospital, Fujian Medical University Carcinoma, Renal Cell; Neoplasms; Lung Neoplasms Details
NP-011 NP-011 Phase 1 Clinical Nexell Therapeutics Inc Myocardial Infarction Details
68Ga-HX01 68GaHX01; 68Ga-HX01 Phase 1 Clinical Hexin (Suzhou) Pharmaceutical Technology Co Ltd Solid tumours; Neoplasms; Contrast agents Details
(68)Ga-RGD Phase 1 Clinical Peking Union Medical College Hospital Keloid Details
fb-PMT NP-100; NP-751 Phase 1 Clinical NanoPharmaceuticals LLC Glioma Details
ACT-50 ACT-50 Phase 1 Clinical Xiamen Amoytop Biotech Co Ltd Neoplasms; Carcinoma, Pancreatic Ductal Details
Pagantangentide Phase 1 Clinical Nanjing Anji Biological Technology Co Ltd, Jiangsu Aotexin Biomedical Technology Co Ltd, China Pharmaceutical University Arthritis, Rheumatoid; Rheumatic Diseases Details

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