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BTK

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Name:Tyrosine-protein kinase BTK
Target Synonym:EC 2.7.10,Bruton S Tyrosine Kinase,IGHD3,EC:2.7.10.2,Tyrosine-protein kinase BTK,AGMX1,ATK,BTK,Bruton Tyrosine Kinase,Bruton Agammaglobulinemia Tyrosine Kinase,B-Cell Progenitor Kinase,Brutons Tyrosine Kinase,BPK,Tyrosine-Protein Kinase BTK Isoform (Lacking Exon 13 To 17),Dominant-Negative Kinase-Deficient Brutons Tyrosine Kinase,Tyrosine-Protein Kinase BTK Isoform (Lacking Exon 14),Truncated Bruton Agammaglobulinemia Tyrosine Kinase,Agammaglobulinaemia Tyrosine Kinase,Agammaglobulinemia Tyrosin
Number of Launched Drugs:6
Number of Drugs in Clinical Trials:64
Lastest Research Phase:Approved

제품 리스트 구매

제품 상태별:
제품 유형별 :
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결합물별:
제품번호 제품 설명 구조 순도 특징
BTK-H55H3 Human Human BTK Protein, His Tag (active enzyme)
BTK-H55H3-structure
BTK-H55H3-sds

공개 약품 정보

Name Research Code Research Phase Company First Brand Name First Approved Country First Indication First Approved Company First Approved Date Indications Clinical Trials
Orelabrutinib ICP-022; BIIB-135 Approved Beijing Innocare Pharma Tech Co Ltd 宜诺凯, INNOBRUKA, YINUOKAI Mainland China Lymphoma, Mantle-Cell; Leukemia, Lymphocytic, Chronic, B-Cell Beijing Innocare Pharma Tech Co Ltd 2020-12-25 Lymphoma, Mantle-Cell; Leukemia, Lymphocytic, Chronic, B-Cell; Central Nervous System Lymphoma; Waldenstrom Macroglobulinemia; Lymphoma; Hepatic Insufficiency; Leukemia, B-Cell; Neuromyelitis Optica; Lupus Erythematosus, Systemic; Multiple Sclerosis, Relapsing-Remitting; Multiple Sclerosis; Lymphoma, Large B-Cell, Diffuse; Arthritis, Rheumatoid; Helicobacter pylori infection; Lymphoma, B-Cell, Marginal Zone; Purpura, Thrombocytopenic, Idiopathic; Lymphoma, B-Cell Details
Ibrutinib PCI-32765; CRA-032765; JNJ-54179060; PCI-32765-00 Approved Pharmacyclics Llc Imbruvica, 亿珂 United States Leukemia, Lymphocytic, Chronic, B-Cell Pharmacyclics Inc 2013-11-13 Waldenstrom Macroglobulinemia; Monoclonal Gammopathy of Undetermined Significance; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Food Hypersensitivity; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Anemia, Aplastic; Prostatic Neoplasms; Leukemia, Prolymphocytic, B-Cell; Hepatic Insufficiency; Leukemia, B-Cell; Lymphoproliferative Disorders; Leukemia, Mast-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Neoplasms, Gonadal Tissue; Intraocular Lymphoma; Lung Neoplasms; Leukemia, Myeloid, Acute; Burkitt Lymphoma; Lymphoma, T-Cell; Central Nervous System Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell; Melanoma; Leukemia, Biphenotypic, Acute; Hepatitis B, Chronic; Leukemia; Skin Melanoma; Lymphoma, B-Cell, Marginal Zone; Immunoproliferative Small Intestinal Disease; Hematopoietic stem cell transplantation (HSCT); Leukemia, Myelogenous, Chronic; HIV Infections; Hematologic Neoplasms; Solid tumours; Carcinoid Tumor; Leukemia, Lymphoid; Esophageal Neoplasms; Lymphoma, B-Cell Details
Acalabrutinib ACP-196 Approved Astrazeneca Plc, Acerta Pharma Llc Calquence, 康可期 United States Lymphoma, Mantle-Cell Astrazeneca Plc 2017-10-31 Multiple Myeloma; Leukemia, Prolymphocytic; Carcinoma, Non-Small-Cell Lung; Central Nervous System Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell; Burkitt Lymphoma; Waldenstrom Macroglobulinemia; Lymphoma; Lymphoma, Non-Hodgkin; Hepatic Insufficiency; Precursor B-Cell Lymphoblastic Leukemia-Lymphoma; Lymphoma, Follicular; Food Hypersensitivity; Richter's Syndrome; Anemia, Hemolytic, Autoimmune; Lymphoma, Mantle-Cell; Drug-Related Side Effects and Adverse Reactions; Pancreatic Neoplasms; Hodgkin Disease; Carcinoma, Transitional Cell; Arthritis, Rheumatoid; Graft vs Host Disease; Neoplasms; Glioblastoma; Coronavirus Disease 2019 (COVID-19); Lymphoma, Large B-Cell, Diffuse; Leukemia, Lymphoid; Squamous Cell Carcinoma of Head and Neck; Leukemia, Hairy Cell; Hematologic Neoplasms; Ovarian Neoplasms; Lymphoma, B-Cell Details
Pirtobrutinib LY 3527727; RXC-005; LOXO-305 Approved Redx Pharma Ltd Jaypirca United States Lymphoma, Mantle-Cell Loxo Oncology Inc 2023-01-27 Purpura, Thrombocytopenic, Idiopathic; Lymphoma, B-Cell, Marginal Zone; Lymphoma, B-Cell; Hematologic Neoplasms; Leukemia; Leukemia, Lymphoid; Renal Insufficiency; Lymphoma, Large B-Cell, Diffuse; Multiple Sclerosis; Multiple Myeloma; Lymphoma, Mantle-Cell; Leukemia, B-Cell; Hepatic Insufficiency; Waldenstrom Macroglobulinemia; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
Tirabrutinib hydrochloride GS-4059; ONO-4059 Approved Ono Pharmaceutical Co Ltd ベレキシブル, Velexbru Japan Lymphoma Ono Pharmaceutical Co Ltd 2020-03-25 Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Sjogren's Syndrome; Chronic Urticaria; Arthritis, Rheumatoid; Lymphoma; Lymphoma, Non-Hodgkin; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell; Pemphigus Details
Zanubrutinib BGB-3111 Approved BeOne Medicines Ltd Brukinsa, 百悦泽 United States Lymphoma, Mantle-Cell Beigene (Usa) Inc 2019-11-14 Lymphoma, Follicular; Carcinoma, Non-Small-Cell Lung; Melanoma; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphohistiocytosis, Hemophagocytic; Lymphoma, T-Cell; Lymphoma; Waldenstrom Macroglobulinemia; Hepatic Insufficiency; Leukemia, B-Cell; Anemia, Hemolytic, Autoimmune; Primary mediastinal B cell lymphoma; Lymphoma, Mantle-Cell; Lymphoma, B-Cell; Lung Diseases; Glomerulonephritis, Membranous; Lupus Nephritis; Neoplasms; Coronavirus Disease 2019 (COVID-19); Lymphoma, Large B-Cell, Diffuse; Immunoglobulin G4-Related Disease; Nephrosis; Leukemia; Solid tumours; Lymphoma, B-Cell, Marginal Zone Details

임상 약품 정보

Name Research Code Research Phase Company Indications Clinical Trials
Nemtabrutinib ARQ-531; MK-1026 Phase 3 Clinical Arqule Inc Hematologic Neoplasms; Lymphoma, B-Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Richter's Syndrome; Hepatic Insufficiency; Waldenstrom Macroglobulinemia; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
Fenebrutinib G-0853; RG-7845; GDC-0853; RO-7010939 Phase 3 Clinical Genentech Inc Arthritis, Rheumatoid; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Lupus Erythematosus, Systemic; Urticaria; Leukemia, Lymphocytic, Chronic, B-Cell Details
Remibrutinib LOU-064; LOU064-NXA; NVP-LOU064-NXA Phase 3 Clinical Novartis Pharma Ag Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Chronic Urticaria; Sjogren's Syndrome; Multiple Sclerosis; Dermatitis; Urticaria; Asthma; Hepatic Insufficiency; Sjogren-Larsson Syndrome; Peanut Hypersensitivity; Hidradenitis Suppurativa; Disease Susceptibility Details
Larotinib Mesylate Z-650 Phase 3 Clinical Guangdong Dongyangguang Pharmaceutical Co Ltd Solid tumours; Esophageal Neoplasms; Pancreatic Neoplasms; Esophageal Squamous Cell Carcinoma Details
Tolebrutinib PRN-2246; SAR-442168 Phase 3 Clinical Principia Biopharma Inc Myasthenia Gravis; Renal Insufficiency; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis; Hepatic Insufficiency Details
Abivertinib A-610MA; AC-0010; AC-0100; AC-001; AC-0010MA; AC-0100-Maleate; EX-ACEA0010MA Phase 3 Clinical Zhejiang Acea Pharmaceutical Co Ltd, Hangzhou Acea Pharmaceutical Research Co Ltd Lymphoma, B-Cell; Coronavirus Disease 2019 (COVID-19); Lymphoma, Large B-Cell, Diffuse; Prostatic Neoplasms; Lymphoma, Mantle-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Carcinoma, Non-Small-Cell Lung; Leukemia, Lymphocytic, Chronic, B-Cell Details
Atuzabrutinib PRN-473; SAR-444727 Phase 2 Clinical Principia Biopharma Inc, Sanofi Dermatitis, Atopic Details
Elsubrutinib/Upadacitinib ABBV-599 Phase 2 Clinical Abbvie Inc Arthritis, Rheumatoid; Lupus Erythematosus, Systemic Details
Poseltinib HM-71224; LY3337641; NB-02 Phase 2 Clinical Hanmi Pharmaceutical Co Ltd Arthritis, Rheumatoid; Lymphoma, Large B-Cell, Diffuse; Central Nervous System Lymphoma; Primary vitreoretinal lymphoma Details
TAS-5315 TAS-5315 Phase 2 Clinical Taiho Pharmaceutical Co Ltd Chronic Urticaria; Arthritis, Rheumatoid Details
HZ-A-018 HZ-A-018 Phase 2 Clinical Hangzhou Yuzheng Pharmaceutical Technology Co Ltd, HeaZen Therapeutics Co Ltd Lymphoma, B-Cell; Multiple Sclerosis; Neuromyelitis Optica; Thrombocytopenia; Central Nervous System Lymphoma Details
Branebrutinib BMS-986195 Phase 2 Clinical Bristol-Myers Squibb Company Arthritis, Rheumatoid; Sjogren's Syndrome; Immune System Diseases; Lupus Erythematosus, Systemic; Dermatitis, Atopic Details
BIIB-091 BIIB-091 Phase 2 Clinical Biogen Inc Multiple Sclerosis, Relapsing-Remitting; Multiple Sclerosis Details
WXFL10230486 WXFL-10230486; WX-486; HWH-486 Phase 2 Clinical Wuxi Apptec Co Ltd, Humanwell Healthcare (Group) Co Ltd Chronic Urticaria; Arthritis, Rheumatoid Details
M-7583 M7583; M-7583 Phase 2 Clinical Merck & Co Inc Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Leukemia, Lymphocytic, Chronic, B-Cell Details
Edralbrutinib TG-1701; SHR-1459 Phase 2 Clinical Jiangsu Hengrui Medicine Co Ltd, Jiangsu shengdi Medicine Co Ltd Lymphoma, B-Cell; Nephrosis; Arthritis, Rheumatoid; Autoimmune Diseases; Glomerulonephritis, Membranous; Neuromyelitis Optica; Lymphoma; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
TL-925 TL-925 Phase 2 Clinical Telios Pharmaceuticals Dry Eye Syndromes; Conjunctivitis, Allergic Details
HBW-3210 HBW-3210; HBW3210 Phase 2 Clinical Chengdu Haibowei Pharmaceutical Co Ltd Lymphoma, B-Cell Details
TQB-3702 TQB3702; TQB-3702 Phase 2 Clinical Jiangsu Chia Tai-Tianqing Pharmaceutical Co Ltd Lymphoma, B-Cell; Hematologic Neoplasms; Neoplasms; Chronic Urticaria; Lupus Erythematosus, Systemic Details
HBW-3220 HBW-3220; HBW-3-10; HBW-003 Phase 2 Clinical Chengdu Haibowei Pharmaceutical Co Ltd Lymphoma, B-Cell; Autoimmune Diseases; Lymphoma, Non-Hodgkin; Glomerulonephritis Details
DZD-8586 DZD-8586 Phase 2 Clinical Dizal (Jiangsu) Pharmaceutical Co Ltd Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
BGB-16673 BGB-16673; [14C]-BGB-16673 Phase 2 Clinical BeOne Medicines Ltd Lymphoma, B-Cell, Marginal Zone; Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Neoplasms; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Leukemia, B-Cell; Lymphoma, Non-Hodgkin; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
HMPL-760 HMPL-760; HMPL760 Phase 2 Clinical Hutchison Medipharma Ltd Lymphoma, B-Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Richter's Syndrome; Lymphoma, Follicular; Lymphoma; Lymphoma, Non-Hodgkin; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
Rocbrutinib LP-168; NWP-775 Phase 2 Clinical Newave Pharmaceutical Inc Lymphoma, B-Cell, Marginal Zone; Hematologic Neoplasms; Lymphoma, B-Cell; Leukemia, Hairy Cell; Neoplasms; Lymphoma, Large B-Cell, Diffuse; Multiple Sclerosis; Neuromyelitis Optica; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
MH-048 MH-048; MH048 Phase 2 Clinical Minghui Pharmaceutical (Shanghai) Co Ltd Lymphoma, B-Cell Details
Elsubrutinib ABBV-105 Phase 2 Clinical Abbvie Ltd Arthritis, Rheumatoid; Lupus Erythematosus, Systemic Details
CX-1440 CX1440; CX-1440 Phase 2 Clinical Hangzhou Sanyintai Pharmaceutical Technology Co Ltd, Hangzhou Aojin Biomedical Technology Co Ltd Lymphoma, B-Cell; Purpura, Thrombocytopenic, Idiopathic; Graft vs Host Disease; Multiple Sclerosis; Lupus Erythematosus, Systemic; Urticaria; Leukemia, B-Cell; Thrombocytopenia Details
JNJ-64264681 JNJ-4681; JNJ-64264681 Phase 1 Clinical Johnson & Johnson Solid tumours; Hematologic Neoplasms; Neoplasms; Myelodysplastic Syndromes; Prostatic Neoplasms, Castration-Resistant; Lymphoma, Non-Hodgkin; Leukemia, Myeloid, Acute; Leukemia, Lymphocytic, Chronic, B-Cell Details
PCI-45292 Phase 1 Clinical Pharmacyclics Llc Arthritis, Rheumatoid; Autoimmune Diseases Details
BMS-935177 Phase 1 Clinical Bristol-Myers Squibb Company Immune System Diseases Details
BT-1053 BT-1053 Phase 1 Clinical Chengdu Brilliant Pharmaceutical Co Ltd, ScinnoHub Pharmaceutical Co Ltd Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell Details
BTK-Max BTK-Max Phase 1 Clinical Bristol-Myers Squibb Company Arthritis, Rheumatoid; Psoriasis Details
DTRMWXHS-12 DTRMWXHS-12; DTRM-12 Phase 1 Clinical Zhejiang Dtrm Biopharma Co Ltd Lymphoma, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell Details
FCN-647 FCN-647 Phase 1 Clinical Fochon Pharmaceuticals Ltd Lymphoma, B-Cell; Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell Details
SN-1011 SN-1011 Phase 1 Clinical Sinomab Bioscience Ltd Lupus Erythematosus, Systemic Details
AC-0058TA AC-0058; AC-0058TA Phase 1 Clinical Hangzhou Acea Pharmaceutical Research Co Ltd, Zhejiang Acea Pharmaceutical Co Ltd Arthritis, Rheumatoid; Lupus Erythematosus, Systemic Details
BI-BTK-1 BI-BTK-1 Phase 1 Clinical C.H. Boehringer Sohn Ag & Co. Kg Lupus Nephritis Details
DTRM-505 DTRM-505 Phase 1 Clinical Lymphoma, B-Cell; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
DWP-212525 DWP-212525 Phase 1 Clinical Daewoong Pharmaceutical Co Ltd Autoimmune Diseases; Arthritis, Rheumatoid; Lupus Erythematosus, Systemic; Pemphigus Details
DWP-213388 DWP-213388 Phase 1 Clinical Daewoong Pharmaceutical Co Ltd Autoimmune Diseases Details
NX-5948 NX-5948 Phase 1 Clinical Nurix Therapeutics Inc Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Follicular; Waldenstrom Macroglobulinemia; Central Nervous System Lymphoma; Leukemia, Lymphocytic, Chronic, B-Cell Details
UBX-303061 UBX-303061 Phase 1 Clinical Ubix Therapeutics Inc Lymphoma, B-Cell Details
[14C]Pirtobrutinib LOXO-305; [14C]RXC-005; RXC-005; [14C]LOXO-305 Phase 1 Clinical Redx Pharma Ltd Details
ANG-0623 ANG-0623; ANG0623 Phase 1 Clinical Angel Pharmaceuticals Co Ltd Multiple Sclerosis Details
XS-04 XS-04 Phase 1 Clinical Jiangsu Xingsheng Xinhui Pharmaceutical Co Ltd Hematologic Neoplasms; Lymphoma, Large B-Cell, Diffuse Details
HZ-Q1070 HZ-Q1070; HZ-Q-1070 Phase 1 Clinical HeaZen Therapeutics Co Ltd Lymphoma, B-Cell; Neoplasms Details
ABBV-101 ABBV-101 Phase 1 Clinical Abbvie Inc Hematologic Neoplasms Details
IMG-004 IMG-004 Phase 1 Clinical Hutchmed (China) Ltd Chronic Urticaria Details
XNW-1011 EVER001; EVER-001; XNW1011; XNW-1011; SN-1011; SN1011 Phase 1 Clinical Suzhou Sinovent Pharmaceuticals Co Ltd, Sinomab Bioscience Ltd Lymphoma, B-Cell; Autoimmune Diseases; Glomerulonephritis, Membranous; Multiple Sclerosis; Neuromyelitis Optica; Lupus Erythematosus, Systemic; Nephrotic Syndrome; Pemphigus Details
AC-0676 AC0676; AC-676; AC676; AC-0676 Phase 1 Clinical Accutar Biotechnology Inc Hematologic Neoplasms; Lymphoma, B-Cell; Autoimmune Diseases Details
JDB175 JDB175 Phase 1 Clinical Shanghai Jiabao Yaoyin Pharmaceutical Technology Co Ltd Lymphoma, Large B-Cell, Diffuse; Multiple Sclerosis Details
SS-001 SS-001 Phase 1 Clinical Zibo Baijichangsheng Pharmaceutical Co Ltd Lymphoma, B-Cell Details
BMS-986196 11C-BMS-986196 Phase 1 Clinical Bristol-Myers Squibb Company Multiple Sclerosis Details
Docirbrutinib AS-1763; BN-102; CB-1763 Phase 1 Clinical Bionova Pharmaceuticals (Shanghai) Ltd, Carna Biosciences Inc Lymphoma, B-Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Leukemia, B-Cell; Waldenstrom Macroglobulinemia; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell Details
Sofnobrutinib AS-0871; AS-871 Phase 1 Clinical Carna Biosciences Inc Autoimmune Diseases Details
NX-2127 NX-2127 Phase 1 Clinical Nurix Therapeutics Inc Lymphoma, B-Cell, Marginal Zone; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Waldenstrom Macroglobulinemia; Leukemia, Lymphocytic, Chronic, B-Cell; Central Nervous System Lymphoma Details
TT-01488 TT-01488 Phase 1 Clinical TransThera Sciences (Nanjing) Inc Lymphoma, B-Cell; Solid tumours; Leukemia, B-Cell Details
SYHA-1811 SYHA-1811 Phase 1 Clinical Shanghai Runshi Pharmaceutical Technology Co Ltd Lymphoma, B-Cell Details
HSK-29116 HSK-29116 Phase 1 Clinical Sichuan Haisco Pharmaceutical Co Ltd Lymphoma, B-Cell Details
YZJ-3058 Phase 1 Clinical Shanghai Haiyan Pharmaceutical Technology Co Ltd Arthritis, Rheumatoid; Lymphoma, Large B-Cell, Diffuse; Leukemia, Lymphocytic, Chronic, B-Cell Details
ZXBT-1158 ZXBT-1158 Phase 1 Clinical Guangzhou BeBetter Medicine Technology Co Lymphoma, B-Cell; Multiple Sclerosis Details
Luxeptinib CG026806; CG-806; CG’806; CG-026806 Phase 1 Clinical Crystalgenomics Inc Hematologic Neoplasms; Myelodysplastic Syndromes; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Follicular; Lymphoma, Non-Hodgkin; Leukemia, Myeloid, Acute; Leukemia, Lymphocytic, Chronic, B-Cell Details
Evobrutinib M-2951; MSC-2364447; MSC-2364447-C; MSC2364447C Phase 1 Clinical Merck Serono Multiple Sclerosis, Relapsing-Remitting; Renal Insufficiency; Arthritis, Rheumatoid; Multiple Sclerosis; Lupus Erythematosus, Systemic; Hepatic Insufficiency Details
GB-5121 GB-5121; GB5121 Clinical Gossamer Bio Inc Neurolymphomatosis; Central Nervous System Lymphoma Details

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