EphA2

EphA2

EphA2 분자 정보

Molecule Name
Ephrin type-A receptor 2
분자 별명
EphA2
Drug Development Progress
임상 약물 수9
시판 약물 수2
최고 연구 개발 단계Approved
표적 별명
EC:2.7.10.1,Epithelial Cell Receptor Protein Tyrosine Kinase,Ephrin type-A receptor 2,Epithelial cell kinase,EPHA2,EPH Receptor A2,Tyrosine-Protein Kinase Receptor ECK,ECK,Soluble EPHA2 Variant 1,EC 2.7.10.1,CTRCT6,ARCC2,CTPP1,CTPA,Receptor, EphA2,EC 2.7.10
분자 배경
Receptor tyrosine kinase which binds promiscuously membrane-bound ephrin-A family ligands residing on adjacent cells, leading to contact-dependent bidirectional signaling into neighboring cells. The signaling pathway downstream of the receptor is referred to as forward signaling while the signaling pathway downstream of the ephrin ligand is referred to as reverse signaling. Activated by the ligand ephrin-A1/EFNA1 regulates migration, integrin-mediated adhesion, proliferation and differentiation of cells. Regulates cell adhesion and differentiation through DSG1/desmoglein-1 and inhibition of the ERK1/ERK2 (MAPK3/MAPK1, respectively) signaling pathway. Engaged by the ligand ephrin-A5/EFNA5 may regulate lens fiber cells shape and interactions and be important for lens transparency development and maintenance. With ephrin-A2/EFNA2 may play a role in bone remodeling through regulation of osteoclastogenesis and osteoblastogenesis.

EphA2 제품 목록

Species
  • Human(2)
  • Rat(1)
Tag
  • His Tag(2)
  • His Tag & Avi Tag(1)
Host
  • HEK293(3)
Conjugate
  • Unconjugated(2)
  • Biotin-labeled(1)
Grade
  • RUO(3)
Low Endotoxin
  • Yes(1)
  • No(2)
분자Cat. No.Product Name종Host구조순도Activity규격 및 가격
EphA2
Human EphA2 Protein, His Tag, low endotoxin (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISA

$230.00

100ug
EphA2
Avitag
EP2-H82E4
Biotinylated Human EphA2 Protein, His,Avitag™ (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISA

$415.00

25ug
EphA2
Rat EphA2 Protein, His Tag (MALS verified)
Rat
HEK293
MALSSDS-PAGE
ELISA

$360.00

100ug
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임상 약물 정보

영어 이름연구 코드연구 개발 단계회사적응증임상 시험
BT-5528BT-5528; BT5528Phase 2 ClinicalBicycle Therapeutics
Carcinoma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Head and Neck Neoplasms; Ovarian Neoplasms; Triple Negative Breast Neoplasms
상세
siRNA-EphA2-DOPCPhase 1 ClinicalThe University Of Texas MD Anderson Cancer Center
Ovarian Neoplasms; Pancreatic Neoplasms; Solid tumours
상세
18F-Dasatinib18F-SKI-249380; [18F]-Fluoro-BMS-354825; [18F]Dasatinib; [18F]SKI-249380; [18F]Fluoro-BMS-354825Phase 1 ClinicalMemorial Sloan Kettering Cancer Center
Bone Marrow Neoplasms; Carcinoma; Diagnostic agents; Lymphoma; Melanoma; Neoplasms; Sarcoma
상세
E-Sync T Cell Therapy (University of California/National Cancer Institute/California Institute for Regenerative Medicine)Phase 1 ClinicalUniversity Of California San Francisco
Glioblastoma
상세
SC-102SC-102Phase 1 ClinicalTianjin Conjustar Biotechnology Co Ltd
Neoplasms; Solid tumours
상세
EphA2-targeted CAR-DCs therapy (Second Affiliated Hospital School Of Zhejiang University School Of Medicine)Phase 1 ClinicalSecond Affiliated Hospital School Of Zhejiang University School Of Medicine
Carcinoma, Non-Small-Cell Lung
상세
EphA2-targeted CAR-T Cells therapy (Second Affiliated Hospital School Of Zhejiang University School Of Medicine)Phase 1 ClinicalSecond Affiliated Hospital School Of Zhejiang University School Of Medicine
Carcinoma, Non-Small-Cell Lung
상세
Autologous Anti-EGFRvIII synNotch Receptor Induced Anti-EphA2/IL-13R alpha2 CAR (E-SYNC) T Cells therapy(California Institute For Regenerative Medicine)Phase 1 ClinicalCalifornia Institute For Regenerative Medicine, National Cancer Institute
Glioblastoma
상세
[18F]AlF-ETN[18F]AlF-ETNPhase 1 ClinicalCapital Medical University, Yunnan Baiyao Group Co Ltd
Prostatic Neoplasms; Solid tumours
상세

시판 약물 정보

영어 이름연구 코드연구 개발 단계회사가장 빠른 브랜드 이름가장 빠른 승인 국가가장 빠른 적응증가장 빠른 승인 회사가장 빠른 승인 날짜적응증임상 시험
RegorafenibDAST; BAY-73-4506ApprovedBayer AGStivarga, ResihanceUnited StatesColorectal NeoplasmsBayer Healthcare Pharmaceuticals Inc2012-09-27
Adenocarcinoma; Adenoma; Bile Duct Neoplasms; Carcinoma, Adenoid Cystic; Carcinoma, Hepatocellular; Carcinoma, Islet Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Ovarian Epithelial; Carcinoma, Renal Cell; Carcinoma, Transitional Cell; Colonic Neoplasms; Colorectal Neoplasms; Esophageal adenocarcinoma; Esophageal Neoplasms; Fallopian Tube Neoplasms; Gastrinoma; Gastrointestinal Neoplasms; Gastrointestinal Stromal Tumors; Glucagonoma; Hemangiosarcoma; Insulinoma; Leukemia, Myeloid, Acute; Liver Neoplasms; Lung Neoplasms; Melanoma; Meningioma; Neoplasm Metastasis; Neoplasms; Osteosarcoma; Ovarian Neoplasms; Pancreatic Neoplasms; Peritoneal Neoplasms; Rectal Neoplasms; Sarcoma; Sarcoma, Ewing; Solid tumours; Somatostatinoma; Stomach Neoplasms; Thymoma; Thyroid Neoplasms
상세
Dasatinib HydrateNSC-732517; BMS-354825ApprovedBristol-Myers Squibb CompanySpraysel, 施达赛, Spricel, SprycelUnited StatesPrecursor Cell Lymphoblastic Leukemia-Lymphoma; Leukemia, Myelogenous, ChronicBristol-Myers Squibb Company2006-06-28
Adenocarcinoma, Clear Cell; Angioimmunoblastic T-cell Lymphoma; Astrocytoma; Blast Crisis; Bone metastases; Brain Neoplasms; Breast Neoplasms; Burkitt Lymphoma; Carcinoma, Basosquamous; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Carcinoma, Verrucous; Cholangiocarcinoma; Chondrosarcoma; Chordoma; Colonic Neoplasms; Coronavirus Disease 2019 (COVID-19); Cystadenocarcinoma; Endometrial Neoplasms; Fallopian Tube Neoplasms; Gastrointestinal Stromal Tumors; Giant Cell Tumor of Bone; Glioblastoma; Glioma; Gliosarcoma; Heart Arrest; Hemangiopericytoma; Hematologic Neoplasms; HIV Infections; Hodgkin Disease; Hormone-Resistant Prostate Neoplasms; Hypereosinophilic Syndrome; Hypopharyngeal Neoplasms; Idiopathic Pulmonary Fibrosis; Immunoproliferative Small Intestinal Disease; Intraocular Lymphoma; Laryngeal Diseases; Laryngeal Neoplasms; Leukemia; Leukemia, Hairy Cell; Leukemia, Large Granular Lymphocytic; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Lymphoid; Leukemia, Myel
상세
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