Thrombopoietin R

Thrombopoietin R

Thrombopoietin R 분자 정보

Molecule Name
Thrombopoietin receptor
분자 별명
MPL,C-MPL,CD110,MPLV,THCYT2,TPOR
Drug Development Progress
임상 약물 수11
시판 약물 수8
최고 연구 개발 단계Approved
표적 별명
CD110 Antigen,THCYT2,C-MPL,CD110,MPLV,Receptors, Thrombopoietin,MPL,TPOR,Myeloproliferative leukemia protein,Myeloproliferative Leukemia Virus Oncogene,Proto-Oncogene C-Mpl,TPO-R,MPL Proto-Oncogene, Thrombopoietin Receptor,Thrombopoietin Receptor,THPOR
분자 배경
Thrombopoietin R, also known as TPO-R, is expressed predominantly on the surface of MKs, platelets, hemangioblasts, and hematopoietic stem cells (HSCs). Binding of TPO to the megakaryocyte TPO-R leads to different effects: prevention of megakaryocyte apoptosis; increased megakaryocyte number, size, and ploidy; increasing rate of megakaryocyte maturation; and internalization of the TPO/TPO-R complex. Thrombopoietin R involved in multiple signal transduction pathways, such as JAK, STAT, and MAP kinase.

Thrombopoietin R 제품 목록

Species
  • Mouse(3)
  • Cynomolgus(2)
  • Porcine(2)
  • Rabbit(2)
  • Human(1)
  • Rat(1)
Tag
  • His Tag(6)
  • His Tag & Avi Tag(5)
Host
  • HEK293(11)
Conjugate
  • Unconjugated(6)
  • Biotin-labeled(5)
Grade
  • RUO(11)
Low Endotoxin
  • Yes(4)
  • No(7)
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임상 약물 정보

영어 이름연구 코드연구 개발 단계회사적응증임상 시험
Romiplostim biosimilar (Enzene Biosciences)267639-76-9Phase 3 ClinicalEnzene Biosciences Ltd
Purpura, Thrombocytopenic, Idiopathic
상세
Romiplostim biosimilar (Intas Pharmaceuticals)Phase 3 ClinicalIntas Biopharmaceuticals
Purpura, Thrombocytopenic, Idiopathic
상세
Romiplostim biosimilar(Generium)GNR-069Phase 3 ClinicalCjsc Generium
Purpura, Thrombocytopenic, Idiopathic
상세
PN-20PN20; PN-20; PJ004; PJ-004Phase 2 ClinicalChongqing Peg-Bio Biopharm Co Ltd
Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
상세
Recombinant human thrombopoietin(Peking University People's Hospital)Phase 2 ClinicalPeking University People'S Hospital
Parturition; Purpura, Thrombocytopenic, Idiopathic
상세
Recombinant human thrombopoietin mimetics (Shandong Quangang)Phase 2 ClinicalShandong Quangang Pharmaceutical Co Ltd
Purpura, Thrombocytopenic, Idiopathic
상세
PEGylated thrombopoietin (Chongqing Paijin Bio)Phase 2 ClinicalChongqing Peg-Bio Biopharm Co Ltd
Hematologic Diseases; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
상세
Romiplostim biosimilar(Geropharma)GP-40141Phase 1 ClinicalGeropharm
Purpura, Thrombocytopenic, Idiopathic
상세
SCB-219SCB-219-M; SCB-219; SCB-219MPhase 1 ClinicalClover Biopharmaceuticals Ltd
Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
상세
Recombinant human thrombopoietin mimetic peptide-Fc fusion protein (Beijing Tide Pharmaceutical)Phase 1 ClinicalBeijing Tide Pharmaceutical Co Ltd
Purpura, Thrombocytopenic, Idiopathic
상세
Thrombopoietin agonist (Scripps Research)3D9ClinicalThe Scripps Research Institute Inc
Thrombocytopenia
상세

시판 약물 정보

영어 이름연구 코드연구 개발 단계회사가장 빠른 브랜드 이름가장 빠른 승인 국가가장 빠른 적응증가장 빠른 승인 회사가장 빠른 승인 날짜적응증임상 시험
Recombinant human thrombopoietin biosimilar (Biolotus)ApprovedBiolotusZypotin-TPOBrazilThrombocytopeniaBiolotus2015-01-01
Thrombocytopenia
상세
RomiplostimAMP-2; AMG-531ApprovedAmgen IncRomiplate, NplateUnited StatesPurpura, Thrombocytopenic, Idiopathic; ThrombocytopeniaAmgen Inc2008-08-22
Acute Radiation Syndrome; Anemia, Aplastic; Bone Marrow Failure Disorders; Carcinoma, Non-Small-Cell Lung; Hematologic Neoplasms; Hodgkin Disease; Lung Neoplasms; Lymphoma; Lymphoma, Non-Hodgkin; Multiple Myeloma; Myelodysplastic Syndromes; Neoplasms; Ovarian Neoplasms; Pancytopenia; Purpura, Thrombocytopenic; Purpura, Thrombocytopenic, Idiopathic; Sarcoma, Ewing; Solid tumours; Thrombocytopenia
상세
LusutrombopagS-888711ApprovedShionogi & Co LtdMulpletaJapanThrombocytopeniaShionogi & Co Ltd2015-09-28
Liver Diseases; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
상세
Herombopag OlamineSHR-8735; SHR 8735 olamineApprovedJiangsu Hengrui Medicine Co LtdHengqu, 恒曲Mainland ChinaAnemia, Aplastic; ThrombocytopeniaJiangsu Hengrui Medicine Co Ltd2021-06-16
Anemia, Aplastic; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Liver Diseases; Lung Neoplasms; Nasopharyngeal Carcinoma; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
상세
Romiplostim biosimilar (Qilu Pharmaceutical)QL-0911ApprovedQilu Pharmaceutical Co Ltd瑞立升Mainland ChinaThrombocytopeniaQilu Pharmaceutical Co Ltd2024-04-02
Anemia, Aplastic; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
상세
Eltrombopag DiolamineSB-497115-GR; ETB-115; SB-497115ApprovedGlaxosmithkline PlcPromacta/Revolade, 瑞弗兰, レボレード, 特艾升, Promacta, RevoladeUnited StatesPurpura, Thrombocytopenic, IdiopathicNovartis Pharma Ag2008-11-20
Anemia, Aplastic; Anemia, Diamond-Blackfan; Blood Platelet Disorders; Bone Marrow Failure Disorders; Bone marrow transplant rejection; Catheter-Related Infections; Delayed Graft Function; Fanconi Anemia; Hematologic Neoplasms; Hematopoietic stem cell transplantation (HSCT); Hemorrhage; Hepatitis B; Hepatitis C; Hepatitis C, Chronic; HIV Infections; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Eosinophilic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myelogenous, Chronic; Leukemia, Myeloid; Leukemia, Myeloid, Accelerated Phase; Leukemia, Myeloid, Acute; Leukemia, Myeloid, Chronic-Phase; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Liver Cirrhosis; Liver Diseases; Metabolic Dysfunction-Associated Steatotic Liver Disease; Multiple Myeloma; Myelodysplastic Syndromes; Neoplasms, Connective and Soft Tissue; Osteosarcoma; Primary Myelofibrosis; Purpura; Purpura, Thrombocytopenic, Id
상세
Avatrombopag MaleateYM-477; AKR-501; AS-1670542; AKR-501-monomaleate; E-5501ApprovedAstellas Pharma Inc苏可欣, Doptelet, DOPTELETUnited StatesThrombocytopenia; Liver DiseasesAkarx Inc2018-05-21
Anemia, Aplastic; Cardiovascular Diseases; Drug-Related Side Effects and Adverse Reactions; Liver Diseases; Lymphoma; Purpura, Thrombocytopenic, Idiopathic; Thrombocytopenia
상세
Recombinant human thrombopoietinrhTPO (3SBio); TPO106; TPO-106ApprovedShenyang Sunshine Pharmaceutical Co Ltd特比奥, Tpiao, 特比澳, TebiaoMainland ChinaThrombocytopenia; Purpura, Thrombocytopenic, IdiopathicShenyang Sunshine Pharmaceutical Co Ltd2005-03-10
Breast Neoplasms; Leukemia; Leukemia, Myeloid, Acute; Liver Cirrhosis; Liver Diseases; Lymphoma; Multiple Myeloma; Myelodysplastic-Myeloproliferative Diseases; Neutropenia; Plasmacytoma; Purpura, Thrombocytopenic, Idiopathic; Radiation sickness; Sepsis; Thrombocytopenia
상세
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