DM-1

DM-1 제품 목록

  • 속성

    Antibody (4)

  • 제품 라이브러리

    온라인 (4)

  • Mouse (3)Rabbit (1)

  • 태그

    - (4)

  • 마커

    Unconjugated (2)HRP Labeled (1)Biotin-labeled (1)

DM-1분자 배경

Mertansine (DM-1) is a tubulin inhibitor that binds to the ends of microtubules and inhibits microtubule dynamics. DM-1(Mertansine) has antitumor activity and functions as a regulator of tubulin. It is an alpha-amino acid ester, a carbamate, an epoxide, an organic heterocyclic tetracyclic compound, an organochlorine compound, a mercaptan, and a maydenin alkaloid. DM-1, derived from Mydenin, is a cytotoxic component of antibody-drug conjugations that produce antibody-drug conjugations via a sulfhydryl group splice with SPP (n-succinimide 4- (2-pyridyl dithio)) or SMCC (4- (3-mercapto-2, 5-dioxy-1 pyrrolidyl) -cyclohexanic acid) splice.

임상 약물 정보

영어 이름연구 코드연구 개발 단계회사적응증임상 시험
Delpacibart eteddesiranAOC-1001; AOC 1001Phase 3 ClinicalAvidity Biosciences IncMyotonic Disorders; Genetic Diseases, Inborn; Musculoskeletal Diseases; Muscular Disorders, Atrophic; Myotonic Dystrophy; Muscular Atrophy; Heredodegenerative Disorders, Nervous System; Muscular Diseases; Neuromuscular Diseases; Nervous System Diseases; Muscular Dystrophies; Neurodegenerative Diseases; Myotonia
상세
Dyne-101Dyne101Phase 2 ClinicalDyne Therapeutics IncMyotonic Dystrophy
상세
ARO-DM1ARO-DM1Phase 2 ClinicalArrowhead Pharmaceuticals IncMyotonic Dystrophy
상세
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  • 임상 약물 정보
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