CNR1

CNR1 분자 정보

영어 이름Cannabinoid CB1 receptor시판 약물 수2
임상 약물 수38표적 별명Cannabinoid Receptor 1 (Brain),CNR1,Cannabinoid Receptor 1,CANN6,CB-R,CNR,CB1,Central Cannabinoid Receptor,CB1K5,CB1A,CB1R,Receptor, Cannabinoid, CB1
최고 연구 개발 단계Approved
영어 이름Cannabinoid CB1 receptor
표적 별명Cannabinoid Receptor 1 (Brain),CNR1,Cannabinoid Receptor 1,CANN6,CB-R,CNR,CB1,Central Cannabinoid Receptor,CB1K5,CB1A,CB1R,Receptor, Cannabinoid, CB1
시판 약물 수2
임상 약물 수38
최고 연구 개발 단계Approved

CNR1 제품 목록

  • 속성

    Protein (3)

  • 제품 라이브러리

    온라인 (3)

  • Human (3)

  • 태그

    - (1)His Tag & Flag Tag (1)His Tag & Avi Tag & Flag Tag (1)

  • 마커

    Unconjugated (2)Biotin-labeled (1)

제품 번호발현 시스템제품 설명단백질 구조순도특성
CN1-H52P6
Human
HEK293
Human CNR1 Full Length Protein (VLP)
CN1-H55D3
Human
InsectCells
Human CNR1 Protein, Flag,His Tag (Detergent)
CN1-H85D3
Human
InsectCells
Biotinylated Human CNR1 Protein, Flag Tag&His,Avitag™ (Detergent)
총 수량3
  • 1

CNR1분자 배경

This gene encodes one of two cannabinoid receptors. The cannabinoids, principally delta-9-tetrahydrocannabinol and synthetic analogs, are psychoactive ingredients of marijuana. The cannabinoid receptors are members of the guanine-nucleotide-binding protein (G-protein) coupled receptor family, which inhibit adenylate cyclase activity in a dose-dependent, stereoselective and pertussis toxin-sensitive manner. The two receptors have been found to be involved in the cannabinoid-induced CNS effects (including alterations in mood and cognition) experienced by users of marijuana. Multiple transcript variants encoding two different protein isoforms have been described for this gene. [provided by RefSeq, May 2009]

CNR1분자 별명

CNR1,cannabinoid receptor 1,CANN6, CB-R, CB1, CB1A, CB1K5, CB1R, CNR

임상 약물 정보

영어 이름연구 코드연구 개발 단계회사적응증임상 시험
Dronabinol(AXIM Biotechnologies)Phase 3 ClinicalAxim Biotechnologies IncAnorexia Nervosa; Cachexia; Child Nutrition Disorders; Nausea; Neoplasms; Nutrition Disorders; Sarcopenia; Vomiting
상세
Cannabidiol soft-gel (Avecho Biotechnology)CBD-TPMPhase 3 ClinicalAvecho Biotechnology LtdSleep Initiation and Maintenance Disorders
상세
Cannabidiol Gel (Zynerba)ZYN002; ZYN-002Phase 3 ClinicalZynerba Pharmaceuticals IncDiGeorge Syndrome; Fragile X Syndrome
상세
AdezunapAP-707Phase 3 ClinicalCannaXan GmbHAccidental Injuries; Back Pain; Brachial Plexus Neuropathies; Brain Injuries, Traumatic; Chronic Pain; Diabetes Mellitus; Diabetic Neuropathies; Diabetic peripheral neuropathy; Low Back Pain; Multiple Sclerosis; Neuralgia; Pain; Pain, Postoperative; Paraplegia; Peripheral Nerve Injuries; Peripheral Nervous System Diseases; Phantom Limb; Somatoform Disorders; Stroke
상세
Dronabinol(Vertanical)VER-01Phase 3 ClinicalVertanical GmbHLow Back Pain
상세
cannabidiol (Cardiol Therapeutics)Phase 3 ClinicalCardiol Therapeutics IncCardiovascular Diseases; Coronavirus Disease 2019 (COVID-19); Myocarditis; Pericarditis
상세
SelonabantV-24343; ANEB-001; VER-24343Phase 2 ClinicalVernalis PlcObesity; Poisoning
상세
11C-MePPEP11C-MePPEPPhase 2 ClinicalEli Lilly And CompanyObesity; Substance-Related Disorders
상세
AX-1602AX-1602Phase 2 ClinicalAxim Biotechnologies IncDermatitis, Atopic; Psoriasis; Vitiligo
상세
NimacimabRYI-018; RYI-028; JNJ-2463Phase 2 ClinicalBird Rock Bio IncDiabetic Gastroparesis; Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity; Renal Insufficiency, Chronic
상세
ART-2713NEO-1940; ART-2713; ART27.13; AZD-1940Phase 2 ClinicalAstrazeneca Plc, Neomed Inc, Pfizer IncAnorexia; Cachexia; Low Back Pain; Pain; Weight Loss
상세
AEF-0217AEF-0217Phase 2 ClinicalAelis FarmaDown Syndrome
상세
MonlunabantS-MRI-1891; (-)-MRI-1891; NN9440–INV-202; INV-202; MRI-1891Phase 2 ClinicalInversago Pharma IncDiabetic Nephropathies; Metabolic Diseases; Metabolic Syndrome; Obesity
상세
Cannabidiol (Ananda Scientific)A-1002-N5S; A1002N5SPhase 2 ClinicalAnanda Scientific IncChronic Pain; Opioid-Related Disorders; Stress Disorders, Post-Traumatic; Tobacco Smoking; Tobacco Use Disorder
상세
Cannabidiol (Biopharmaceutical Research Company)BRC-001Phase 2 ClinicalBiopharmaceutical Research CompanyBreast Neoplasms; Carcinoma, Ductal, Breast
상세
C20T5C20T5Phase 2 ClinicalMurdoch Childrens Research Institute
상세
C12T12C12T12Phase 2 ClinicalMurdoch Childrens Research Institute
상세
SuvadronabinolTHC-VHS-NEC; SBI-100; NB-1111; Sb-100 OE; SBI-100 OE; THCVHS; THCVHS-N; THCVHS-NE; UM-5050Phase 2 ClinicalUniversity Of MississippiGlaucoma; Glaucoma, Open-Angle; Ocular Hypertension
상세
IGC-AD1IGC-AD1Phase 2 ClinicalUniversity Of South FloridaAlzheimer Disease; Dementia; Psychomotor Agitation
상세
LixosiconeAEF-0117Phase 2 ClinicalAelis Farma, National Institute On Drug AbuseMarijuana Abuse
상세
ZYN-001ZYN-001Phase 1 ClinicalZynerba PharmaceuticalsFibromyalgia; Neuralgia
상세
TetrahydrocannabivarinGWP-42004; THCV; O-4394; DELTA9-THCV; GW-42004Phase 1 ClinicalGw Pharmaceuticals PlcDiabetes Mellitus, Type 2; Dyslipidemias; Hypercholesterolemia; Hyperglycemia; Metabolic Syndrome; Obesity, Morbid
상세
Cannabidiol/hydroxychloroquineIHL-675A; IHL-675Phase 1 ClinicalIncannex Healthcare LtdArthritis, Rheumatoid; Respiratory Distress Syndrome, Adult
상세
ZevaquenabantMRI-1867; (S)-MRI-1867; INV-101Phase 1 ClinicalNational Institutes Of HealthScleroderma, Systemic
상세
Cannabidiol (Artelo Biosciences)ART-12.11; ART12.11; ART-1211Phase 1 ClinicalArtelo Biosciences IncAnxiety; Depression; Depressive Disorder
상세
S1-221S1-221Phase 1 ClinicalDelphian Therapeutics Australia Pty Ltd
상세
Cannabidiol (Tiamat Australia)MRX-1Phase 1 ClinicalTiamat Australia Pty Ltd
상세
Atorvastatin Calcium Hydrate/CannabidiolPhase 1 ClinicalIndication Bioscience LLCCoronary Disease; Dyslipidemias
상세
TPT0301TPT-0301; TPT0301Phase 1 ClinicalTetra Pharm Technologies ApSChronic Pain
상세
INV-347NN9441; NN-9441; INV-347Phase 1 ClinicalInversago Pharma IncObesity
상세
IPI 201(Isosceles Pharmaceuticals Inc )IPI-201Phase 1 ClinicalPain, Postoperative
상세
CRB-913CRB-913Phase 1 ClinicalJenrin Discovery LLCObesity
상세
GFB-024Phase 1 ClinicalTakeda PharmaDiabetes Complications; Diabetes Mellitus; Diabetic Nephropathies; Endocrine System Diseases; Kidney Diseases
상세
DBPR-211Phase 1 ClinicalNational Health Research InstitutesDiabetes Mellitus, Type 2
상세
MP-10XMP-10XClinicalMedipure HoldingsPain
상세
MP-20XMP-20XClinicalMedipure HoldingsAnxiety Disorders; Mood Disorders
상세
Cannabidiol (Receptor Life Sciences)ClinicalReceptor Life Sciences IncAutism Spectrum Disorder
상세
Cannabidiol/PalmitoylethanolamideSCI–210; THX-210ClinicalTherapix Biosciences LtdAutism Spectrum Disorder; Diabetic Neuropathies
상세

시판 약물 정보

영어 이름연구 코드연구 개발 단계회사가장 빠른 브랜드 이름가장 빠른 승인 국가가장 빠른 적응증가장 빠른 승인 회사가장 빠른 승인 날짜적응증임상 시험
Cannabidiol/Dronabinoldelta-9-THC/CBD; MPL-001; MPL-005; PPP-011; BOL-DP-o-04; GW-1000-02; PPP-001; MGC-ODT; GW-1000; KL16-012; THC-5ApprovedGw PharmaceuticalsSativex, Qixleef, QIXLEEFTMCanadaCancer Pain; Chronic Pain; Muscle Spasticity; Neuralgia; Multiple Sclerosisnull2005-04-01Acute Pain; Agitation; Agoraphobia; Anorexia; Anxiety Disorders; Arthritis, Psoriatic; Arthritis, Rheumatoid; Back Pain; Cancer Pain; Cerebral Palsy; Chronic Pain; Corticobasal degeneration; Dementia; Depression; Depressive Disorder, Major; Diabetic Neuropathies; Drug Resistant Epilepsy; Essential Tremor; Genital Diseases, Male; Healthy Aging; Hepatic Insufficiency; Hidradenitis Suppurativa; Huntington Disease; Kidney Diseases; Low Back Pain; Malnutrition; Marijuana Abuse; Marijuana Use; Migraine Disorders; Multiple Sclerosis; Muscle Spasticity; Neck Pain; Neoplasms; Neuralgia; Neuralgia, Postherpetic; Neuromyelitis Optica; Opioid-Related Disorders; Osteoarthritis, Knee; Pain; Panic Disorder; Peripheral Nervous System Diseases; Phobia, Social; Psoriasis; Reflex Sympathetic Dystrophy; Renal Insufficiency; Renal Insufficiency, Chronic; Sciatica; Sleep Initiation and Maintenance Disorders; Sleep Wake Disorders; Social Behavior; Spasm; Spinal Cord Injuries; Squamous Cell Carcinoma of Head and Neck; Stress Disorde
상세
CannabidiolCHI-902; APH-1501; GLA-015; BTX-1503; BTX-1801; GWP-42003-P; BOL-DP-o-05; GW-42003; BTX-1204; PTL-101; BTX-1702; PBX-1308; BRCX-014; LYT-310; GWP-42003ApprovedGw Pharmaceuticals PlcEpidyolex, Cannepil, EpidiolexUnited StatesEpilepsies, Myoclonic; Lennox Gastaut Syndromenull2018-06-25Acne Vulgaris; Acute Pain; Alcohol Abstinence; Alcoholic Intoxication; Alcoholism; Anemia, Sickle Cell; Anorexia Nervosa; Anxiety; Anxiety Disorders; Appetitive Behavior; Arthralgia; Arthritis, Psoriatic; Arthritis, Rheumatoid; Autism Spectrum Disorder; Autistic Disorder; Azotemia; Behavior, Addictive; Bipolar Disorder; Blepharospasm; Brain Diseases; Brain Injuries, Traumatic; Breast Neoplasms; Bruxism; Burnout, Psychological; Cachexia; Carcinoma, Non-Small-Cell Lung; Carpal Tunnel Syndrome; Central Nervous System Diseases; Child Behavior Disorders; Chronic Pain; Chronic Periodontitis; Chronic Urticaria; Cicatrix; Cognition Disorders; Cognitive Dysfunction; Colitis, Ulcerative; Colorectal Neoplasms; Coronavirus Disease 2019 (COVID-19); Corticobasal degeneration; Craving; Crohn Disease; Cystitis, Interstitial; Dentin Sensitivity; Depression; Dermatitis, Atopic; Diabetes Mellitus, Type 2; Diabetic Neuropathies; Driving Under the Influence; Drug Resistant Epilepsy; Dyslipidemias; Dysmenorrhea; Dyspepsia; Eczema;
상세
  • 분자 정보
  • 제품 목록
  • 시판 약물 정보
  • 임상 약물 정보
문의하기

전화
글로벌: +1 800-810-0816 (무료)
아시아태평양: +86 400-682-2521

주소 서울특별시 송파구 법원로11길 11, 제3층 제비-314,315호