CNR1

CNR1

CNR1 분자 정보

Molecule Name
Cannabinoid CB1 receptor
분자 별명
CNR1,cannabinoid receptor 1,CANN6, CB-R, CB1, CB1A, CB1K5, CB1R, CNR
Drug Development Progress
임상 약물 수38
시판 약물 수2
최고 연구 개발 단계Approved
표적 별명
Cannabinoid Receptor 1 (Brain),CNR1,Cannabinoid Receptor 1,CANN6,CB-R,CNR,CB1,Central Cannabinoid Receptor,CB1K5,CB1A,CB1R,Receptor, Cannabinoid, CB1
분자 배경
This gene encodes one of two cannabinoid receptors. The cannabinoids, principally delta-9-tetrahydrocannabinol and synthetic analogs, are psychoactive ingredients of marijuana. The cannabinoid receptors are members of the guanine-nucleotide-binding protein (G-protein) coupled receptor family, which inhibit adenylate cyclase activity in a dose-dependent, stereoselective and pertussis toxin-sensitive manner. The two receptors have been found to be involved in the cannabinoid-induced CNS effects (including alterations in mood and cognition) experienced by users of marijuana. Multiple transcript variants encoding two different protein isoforms have been described for this gene.

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임상 약물 정보

영어 이름연구 코드연구 개발 단계회사적응증임상 시험
Dronabinol(AXIM Biotechnologies)Phase 3 ClinicalAxim Biotechnologies Inc
Anorexia Nervosa; Cachexia; Child Nutrition Disorders; Nausea; Neoplasms; Nutrition Disorders; Sarcopenia; Vomiting
상세
Cannabidiol soft-gel (Avecho Biotechnology)CBD-TPMPhase 3 ClinicalAvecho Biotechnology Ltd
Sleep Initiation and Maintenance Disorders
상세
Cannabidiol Gel (Zynerba)ZYN002; ZYN-002Phase 3 ClinicalZynerba Pharmaceuticals Inc
DiGeorge Syndrome; Fragile X Syndrome
상세
AdezunapAP-707Phase 3 ClinicalCannaXan GmbH
Accidental Injuries; Back Pain; Brachial Plexus Neuropathies; Brain Injuries, Traumatic; Chronic Pain; Diabetes Mellitus; Diabetic Neuropathies; Diabetic peripheral neuropathy; Low Back Pain; Multiple Sclerosis; Neuralgia; Pain; Pain, Postoperative; Paraplegia; Peripheral Nerve Injuries; Peripheral Nervous System Diseases; Phantom Limb; Somatoform Disorders; Stroke
상세
Dronabinol(Vertanical)VER-01Phase 3 ClinicalVertanical GmbH
Low Back Pain
상세
cannabidiol (Cardiol Therapeutics)Phase 3 ClinicalCardiol Therapeutics Inc
Cardiovascular Diseases; Coronavirus Disease 2019 (COVID-19); Myocarditis; Pericarditis
상세
SelonabantV-24343; ANEB-001; VER-24343Phase 2 ClinicalVernalis Plc
Obesity; Poisoning
상세
11C-MePPEP11C-MePPEPPhase 2 ClinicalEli Lilly And Company
Obesity; Substance-Related Disorders
상세
AX-1602AX-1602Phase 2 ClinicalAxim Biotechnologies Inc
Dermatitis, Atopic; Psoriasis; Vitiligo
상세
NimacimabRYI-018; RYI-028; JNJ-2463Phase 2 ClinicalBird Rock Bio Inc
Diabetic Gastroparesis; Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity; Renal Insufficiency, Chronic
상세
ART-2713NEO-1940; ART-2713; ART27.13; AZD-1940Phase 2 ClinicalAstrazeneca Plc, Neomed Inc, Pfizer Inc
Anorexia; Cachexia; Low Back Pain; Pain; Weight Loss
상세
AEF-0217AEF-0217Phase 2 ClinicalAelis Farma
Down Syndrome
상세
MonlunabantS-MRI-1891; (-)-MRI-1891; NN9440–INV-202; INV-202; MRI-1891Phase 2 ClinicalInversago Pharma Inc
Diabetic Nephropathies; Metabolic Diseases; Metabolic Syndrome; Obesity
상세
Cannabidiol (Ananda Scientific)A-1002-N5S; A1002N5SPhase 2 ClinicalAnanda Scientific Inc
Chronic Pain; Opioid-Related Disorders; Stress Disorders, Post-Traumatic; Tobacco Smoking; Tobacco Use Disorder
상세
Cannabidiol (Biopharmaceutical Research Company)BRC-001Phase 2 ClinicalBiopharmaceutical Research Company
Breast Neoplasms; Carcinoma, Ductal, Breast
상세
C20T5C20T5Phase 2 ClinicalMurdoch Childrens Research Institute
상세
C12T12C12T12Phase 2 ClinicalMurdoch Childrens Research Institute
상세
SuvadronabinolTHC-VHS-NEC; SBI-100; NB-1111; Sb-100 OE; SBI-100 OE; THCVHS; THCVHS-N; THCVHS-NE; UM-5050Phase 2 ClinicalUniversity Of Mississippi
Glaucoma; Glaucoma, Open-Angle; Ocular Hypertension
상세
IGC-AD1IGC-AD1Phase 2 ClinicalUniversity Of South Florida
Alzheimer Disease; Dementia; Psychomotor Agitation
상세
LixosiconeAEF-0117Phase 2 ClinicalAelis Farma, National Institute On Drug Abuse
Marijuana Abuse
상세
ZYN-001ZYN-001Phase 1 ClinicalZynerba Pharmaceuticals
Fibromyalgia; Neuralgia
상세
TetrahydrocannabivarinGWP-42004; THCV; O-4394; DELTA9-THCV; GW-42004Phase 1 ClinicalGw Pharmaceuticals Plc
Diabetes Mellitus, Type 2; Dyslipidemias; Hypercholesterolemia; Hyperglycemia; Metabolic Syndrome; Obesity, Morbid
상세
Cannabidiol/hydroxychloroquineIHL-675A; IHL-675Phase 1 ClinicalIncannex Healthcare Ltd
Arthritis, Rheumatoid; Respiratory Distress Syndrome, Adult
상세
ZevaquenabantMRI-1867; (S)-MRI-1867; INV-101Phase 1 ClinicalNational Institutes Of Health
Scleroderma, Systemic
상세
Cannabidiol (Artelo Biosciences)ART-12.11; ART12.11; ART-1211Phase 1 ClinicalArtelo Biosciences Inc
Anxiety; Depression; Depressive Disorder
상세
S1-221S1-221Phase 1 ClinicalDelphian Therapeutics Australia Pty Ltd
상세
Cannabidiol (Tiamat Australia)MRX-1Phase 1 ClinicalTiamat Australia Pty Ltd
상세
Atorvastatin Calcium Hydrate/CannabidiolPhase 1 ClinicalIndication Bioscience LLC
Coronary Disease; Dyslipidemias
상세
TPT0301TPT-0301; TPT0301Phase 1 ClinicalTetra Pharm Technologies ApS
Chronic Pain
상세
INV-347NN9441; NN-9441; INV-347Phase 1 ClinicalInversago Pharma Inc
Obesity
상세
IPI 201(Isosceles Pharmaceuticals Inc )IPI-201Phase 1 Clinical
Pain, Postoperative
상세
CRB-913CRB-913Phase 1 ClinicalJenrin Discovery LLC
Obesity
상세
GFB-024Phase 1 ClinicalTakeda Pharma
Diabetes Complications; Diabetes Mellitus; Diabetic Nephropathies; Endocrine System Diseases; Kidney Diseases
상세
DBPR-211Phase 1 ClinicalNational Health Research Institutes
Diabetes Mellitus, Type 2
상세
MP-10XMP-10XClinicalMedipure Holdings
Pain
상세
MP-20XMP-20XClinicalMedipure Holdings
Anxiety Disorders; Mood Disorders
상세
Cannabidiol (Receptor Life Sciences)ClinicalReceptor Life Sciences Inc
Autism Spectrum Disorder
상세
Cannabidiol/PalmitoylethanolamideSCI–210; THX-210ClinicalTherapix Biosciences Ltd
Autism Spectrum Disorder; Diabetic Neuropathies
상세

시판 약물 정보

영어 이름연구 코드연구 개발 단계회사가장 빠른 브랜드 이름가장 빠른 승인 국가가장 빠른 적응증가장 빠른 승인 회사가장 빠른 승인 날짜적응증임상 시험
Cannabidiol/Dronabinoldelta-9-THC/CBD; MPL-001; MPL-005; PPP-011; BOL-DP-o-04; GW-1000-02; PPP-001; MGC-ODT; GW-1000; KL16-012; THC-5ApprovedGw PharmaceuticalsSativex, Qixleef, QIXLEEFTMCanadaCancer Pain; Chronic Pain; Muscle Spasticity; Neuralgia; Multiple Sclerosisnull2005-04-01
Acute Pain; Agitation; Agoraphobia; Anorexia; Anxiety Disorders; Arthritis, Psoriatic; Arthritis, Rheumatoid; Back Pain; Cancer Pain; Cerebral Palsy; Chronic Pain; Corticobasal degeneration; Dementia; Depression; Depressive Disorder, Major; Diabetic Neuropathies; Drug Resistant Epilepsy; Essential Tremor; Genital Diseases, Male; Healthy Aging; Hepatic Insufficiency; Hidradenitis Suppurativa; Huntington Disease; Kidney Diseases; Low Back Pain; Malnutrition; Marijuana Abuse; Marijuana Use; Migraine Disorders; Multiple Sclerosis; Muscle Spasticity; Neck Pain; Neoplasms; Neuralgia; Neuralgia, Postherpetic; Neuromyelitis Optica; Opioid-Related Disorders; Osteoarthritis, Knee; Pain; Panic Disorder; Peripheral Nervous System Diseases; Phobia, Social; Psoriasis; Reflex Sympathetic Dystrophy; Renal Insufficiency; Renal Insufficiency, Chronic; Sciatica; Sleep Initiation and Maintenance Disorders; Sleep Wake Disorders; Social Behavior; Spasm; Spinal Cord Injuries; Squamous Cell Carcinoma of Head and Neck; Stress Disorde
상세
CannabidiolCHI-902; APH-1501; GLA-015; BTX-1503; BTX-1801; GWP-42003-P; BOL-DP-o-05; GW-42003; BTX-1204; PTL-101; BTX-1702; PBX-1308; BRCX-014; LYT-310; GWP-42003ApprovedGw Pharmaceuticals PlcEpidyolex, Cannepil, EpidiolexUnited StatesEpilepsies, Myoclonic; Lennox Gastaut Syndromenull2018-06-25
Acne Vulgaris; Acute Pain; Alcohol Abstinence; Alcoholic Intoxication; Alcoholism; Anemia, Sickle Cell; Anorexia Nervosa; Anxiety; Anxiety Disorders; Appetitive Behavior; Arthralgia; Arthritis, Psoriatic; Arthritis, Rheumatoid; Autism Spectrum Disorder; Autistic Disorder; Azotemia; Behavior, Addictive; Bipolar Disorder; Blepharospasm; Brain Diseases; Brain Injuries, Traumatic; Breast Neoplasms; Bruxism; Burnout, Psychological; Cachexia; Carcinoma, Non-Small-Cell Lung; Carpal Tunnel Syndrome; Central Nervous System Diseases; Child Behavior Disorders; Chronic Pain; Chronic Periodontitis; Chronic Urticaria; Cicatrix; Cognition Disorders; Cognitive Dysfunction; Colitis, Ulcerative; Colorectal Neoplasms; Coronavirus Disease 2019 (COVID-19); Corticobasal degeneration; Craving; Crohn Disease; Cystitis, Interstitial; Dentin Sensitivity; Depression; Dermatitis, Atopic; Diabetes Mellitus, Type 2; Diabetic Neuropathies; Driving Under the Influence; Drug Resistant Epilepsy; Dyslipidemias; Dysmenorrhea; Dyspepsia; Eczema;
상세